Mihaela-Liliana Ţînţaş

Donepezil-Based Central Acetylcholinesterase Inhibitors by Means of a “Bio-Oxidizable” Prodrug Strategy: Design, Synthesis, and in Vitro Biological Evaluation

Ludovic Peauger, Rabah Azzouz, Vincent Gembus et al. · Journal of Medicinal Chemistry · 2017 · 93 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

An Overview of the Synthesis of Highly Versatile N-Hydroxysuccinimide Esters

Cyril Papamicaël, Vincent Gembus, Anaïs Barré et al. · Synthesis · 2016 · 47 citations

Pharmacy, Biochemistry, Bioorganic Chemistry +6

Novel donepezil-like N-benzylpyridinium salt derivatives as AChE inhibitors and their corresponding dihydropyridine “bio-oxidizable” prodrugs: Synthesis, biological evaluation and structure-activity relationship

Rabah Azzouz, Ludovic Peauger, Vincent Gembus et al. · European Journal of Medicinal Chemistry · 2017 · 39 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Palladium-Catalyzed Carbonylation of (Hetero)Aryl, Alkenyl and Allyl Halides by Means of <i>N-</i>Hydroxysuccinimidyl Formate as CO Surrogate

Anaïs Barré, Mihaela-Liliana Ţînţaş, Florent Alix et al. · The Journal of Organic Chemistry · 2015 · 33 citations

Natural Sciences, Chemistry, Catalysis +16

Dihydroquinoline Carbamate Derivatives as “Bio-oxidizable” Prodrugs for Brain Delivery of Acetylcholinesterase Inhibitors: [¹¹C] Radiosynthesis and Biological Evaluation

Pierre Bohn, Fabienne Gourand, Cyril Papamicaël et al. · ACS Chemical Neuroscience · 2015 · 32 citations

Pharmacy, Medicinal Chemistry, Pharmacology +14