Concepedia
Statistics
Publications
11
Citations
552
H-Index
Active since
2017
Affiliations
University of Bonn(Current)
Leipzig University
Shandong University
Saint Louis University
City University of Hong Kong, Shenzhen Research Institute
Katharina Sylvester is an author at University of Bonn specializing in drug discovery, medicinal chemistry, and natural sciences.
Top concepts
MedicineBiochemistryGlycobiologyPharmacologyCell SignalingDrug DiscoveryChemical BiologyNatural SciencesMedicinal ChemistrySignal Transduction
Publications per year
2017–2024
Targeting the Main Protease of SARS‐CoV‐2: From the Establishment of High Throughput Screening to the Design of Tailored Inhibitors
Julian Breidenbach, Carina Lemke, Thanigaimalai Pillaiyar et al. · Angewandte Chemie International Edition · 2021 · 143 citations · Full text
Diindolylmethane Derivatives: Potent Agonists of the Immunostimulatory Orphan G Protein-Coupled Receptor GPR84
Thanigaimalai Pillaiyar, Meryem Köse, Katharina Sylvester et al. · Journal of Medicinal Chemistry · 2017 · 97 citations · Full text
Discovery and Crystallographic Studies of Trisubstituted Piperazine Derivatives as Non-Covalent SARS-CoV-2 Main Protease Inhibitors with High Target Specificity and Low Toxicity
Shenghua Gao, Katharina Sylvester, Letian Song et al. · Journal of Medicinal Chemistry · 2022 · 78 citations · Full text
Small-Molecule Thioesters as SARS-CoV-2 Main Protease Inhibitors: Enzyme Inhibition, Structure–Activity Relationships, Antiviral Activity, and X-ray Structure Determination
Thanigaimalai Pillaiyar, Philipp Flury, Nadine Krüger et al. · Journal of Medicinal Chemistry · 2022 · 66 citations · Full text
6-(Ar)Alkylamino-Substituted Uracil Derivatives: Lipid Mimetics with Potent Activity at the Orphan G Protein-Coupled Receptor 84 (GPR84)
Thanigaimalai Pillaiyar, Meryem Köse, Vigneshwaran Namasivayam et al. · ACS Omega · 2018 · 37 citations · Full text
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