Freddy Rivault

The synthesis and biological evaluation of novel series of nitrile-containing fluoroquinolones as antibacterial agents

Sean T. Murphy, Heather L. Case, Edmund L. Ellsworth et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 88 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Tyrosine Kinase Inhibitors. 20. Optimization of Substituted Quinazoline and Pyrido[3,4-<i>d</i>]pyrimidine Derivatives as Orally Active, Irreversible Inhibitors of the Epidermal Growth Factor Receptor Family

Jeff B. Smaill, Andrea J. Gonzales, Julie A. Spicer et al. · Journal of Medicinal Chemistry · 2016 · 60 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Synthesis and biological evaluation of the suberoylanilide hydroxamic acid (SAHA) β-glucuronide and β-galactoside for application in selective prodrug chemotherapy

Mickaël Thomas, Freddy Rivault, Isabelle Tranoy‐Opalinski et al. · Bioorganic & Medicinal Chemistry Letters · 2006 · 40 citations

Pharmacy, Medicinal Chemistry, Pharmacology +10

Synthesis of functionalized analogs of pyochelin, a siderophore of Pseudomonas aeruginosa and Burkholderia cepacia

Freddy Rivault, Viviane Schons, Clémence Liébert et al. · Tetrahedron · 2005 · 21 citations

Life Sciences, Microbiology, Bioorganic Chemistry +4

Synthesis and biological properties of iron chelators based on a bis-2-(2-hydroxy-phenyl)-thiazole-4-carboxamide or -thiocarboxamide (BHPTC) scaffold

David Rodríguez‐Lucena, François Gaboriau, Freddy Rivault et al. · Bioorganic & Medicinal Chemistry · 2009 · 18 citations

Natural Sciences, Chemistry, Medicinal Chemistry +13