Stephacidin A and B:  Two Structurally Novel, Selective Inhibitors of the Testosterone-Dependent Prostate LNCaP Cells

Jingfang Qian‐Cutrone, Stella Huang, Yue‐Zhong Shu, +7

Journal of the American Chemical Society

Secondary MetaboliteSelective InhibitorsPharmacotherapyNovel AlkaloidsPharmaceutical Chemistry +17

Synthesis and Structure−Activity Relationships of 3-Aryloxindoles:  A New Class of Calcium-Dependent, Large Conductance Potassium (Maxi-K) Channel Openers with Neuroprotective Properties

Piyasena Hewawasam, Matthew Erway, Sandra L. Moon, +8

Journal of Medicinal Chemistry

Xenopus LaevisChemistryChemical BiologyLarge Conductance PotassiumHyperpolarization (Biology) +14

The synthesis and characterization of BMS-204352 (MaxiPost™) and related 3-fluorooxindoles as openers of maxi-K potassium channels

Piyasena Hewawasam, Valentin K. Gribkoff, Yadagiri Pendri, +12

Bioorganic & Medicinal Chemistry Letters

Materials ScienceRelated 3-FluorooxindolesMaxi-k Potassium ChannelsChemistry

The Impact of Palladium(II) Reduction Pathways on the Structure and Activity of Palladium(0) Catalysts

Carolyn S. Wei, Geraint H. M. Davies, Omid Soltani, +6

Angewandte Chemie International Edition

Materials ScienceInorganic ChemistryChemical EngineeringEngineeringReduction Pathways +10

Enantioselective Synthesis of a Highly Potent Selective Serotonin Reuptake Inhibitor. An Application of Imidazolidinone Catalysis to the Alkylation of Indoles with an α,β-Disubstituted α,β-Unsaturated Aldehyde

Dalton King, Zhaoxing Meng, Derek J. Denhart, +5

Organic Letters

Asymmetric CatalysisMedicinal ChemistryEnantioselective SynthesisImidazolidinone Catalyst 3BNatural Sciences +13

The Discovery of Asunaprevir (BMS-650032), An Orally Efficacious NS3 Protease Inhibitor for the Treatment of Hepatitis C Virus Infection

Paul M. Scola, Li‐Qiang Sun, Alan Xiangdong Wang, +47

Journal of Medicinal Chemistry

Inhibitors of Human Immunodeficiency Virus Type 1 (HIV-1) Attachment. 5. An Evolution from Indole to Azaindoles Leading to the Discovery of 1-(4-Benzoylpiperazin-1-yl)-2-(4,7-dimethoxy-1<i>H</i>-pyrrolo[2,3-<i>c</i>]pyridin-3-yl)ethane-1,2-dione (BMS-488043), a Drug Candidate That Demonstrates Antiviral Activity in HIV-1-Infected Subjects

Tao Wang, Zhiwei Yin, Zhongxing Zhang, +23

Journal of Medicinal Chemistry

Organic ChemistryHiv-1-infected SubjectsPharmacotherapyAntiviral DrugAzaindole Leads +17

Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase

Robert G. Gentles, Min Ding, John A. Bender, +43

Journal of Medicinal Chemistry

Structure of the pure-spermine form of Z-DNA (magnesium free) at 1-.ANG. resolution

Martin Egli, Loren Dean Williams, Qi Gao, +1

Biochemistry

SpermatogenesisInorganic ChemistryX-ray CrystallographyDna Hexamer DCrystal Structure +13

Amorphous Drug-PVP Dispersions: Application of Theoretical, Thermal and Spectroscopic Analytical Techniques to the Study of a Molecule With Intermolecular Bonds in Both the Crystalline and Pure Amorphous State

Jonathan Brown, Andrew B. Dennis, M. Fakes, +8

Journal of Pharmaceutical Sciences

Materials ScienceEngineeringPolymer SolutionPolymer SciencePhysical Chemistry +7