Caroline Denevault‐Sabourin

Structure-based design of novel quinoxaline-2-carboxylic acids and analogues as Pim-1 inhibitors

Bruno Oyallon, Marie Brachet‐Botineau, Cédric Logé et al. · European Journal of Medicinal Chemistry · 2018 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Development of new highly potent imidazo[1,2-b]pyridazines targeting Toxoplasma gondii calcium-dependent protein kinase 1

Espérance Moine, Isabelle Dimier‐Poisson, Cécile Enguehard‐Gueiffier et al. · European Journal of Medicinal Chemistry · 2015 · 28 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

A small-molecule cell-based screen led to the identification of biphenylimidazoazines with highly potent and broad-spectrum anti-apicomplexan activity

Espérance Moine, Caroline Denevault‐Sabourin, Françoise Debierre-Grockiego et al. · European Journal of Medicinal Chemistry · 2014 · 22 citations

Pharmacy, Chemistry, Medicinal Chemistry +8

New Quinoxaline Derivatives as Dual Pim-1/2 Kinase Inhibitors: Design, Synthesis and Biological Evaluation

Bruno Oyallon, Marie Brachet‐Botineau, Cédric Logé et al. · Molecules · 2021 · 21 citations · Full text

Medicine, Medicinal Chemistry, Oncology +12

Branched pegylated linker-auristatin to control hydrophobicity for the production of homogeneous minibody-drug conjugate against HER2-positive breast cancer

Emmanuel Douez, Émilie Allard-Vannier, Imène Ait Mohamed Amar et al. · Journal of Controlled Release · 2024 · 21 citations

Pharmacy, Oncology, Pharmacology +14