Concepedia
Statistics
Publications
16
Citations
516
H-Index
14
Active since
2010
Affiliations
Shanghai Institute of Materia Medica(Current)
Chinese Academy of Sciences
University of Chinese Academy of Sciences
Shanghai Institute of Applied Physics
Shanghai Institute of Pharmaceutical Industry
Yanlian Li is an author at Shanghai Institute of Materia Medica specializing in medicine, drug discovery, and pharmacology.
Top concepts
MedicineDrug DiscoveryPharmacologyBiochemistryDrug DevelopmentNatural SciencesChemical BiologyMedicinal ChemistryPharmacotherapyMolecular Biology
Publications per year
2010–2024
Fragment-Based Drug Discovery of 2-Thiazolidinones as Inhibitors of the Histone Reader BRD4 Bromodomain
Lele Zhao, Danyan Cao, Tiantian Chen et al. · Journal of Medicinal Chemistry · 2013 · 118 citations · Full text
Molecular Docking, Fragment 8, Medicinal Chemistry +14
Fragment-Based Drug Discovery of 2-Thiazolidinones as BRD4 Inhibitors: 2. Structure-Based Optimization
Lele Zhao, Ying-Qing Wang, Danyan Cao et al. · Journal of Medicinal Chemistry · 2015 · 49 citations · Full text
Structure-Based Discovery and Development of a Series of Potent and Selective Bromodomain and Extra-Terminal Protein Inhibitors
Jianping Hu, Changqing Tian, Mohammadali Soleimani Damaneh et al. · Journal of Medicinal Chemistry · 2019 · 37 citations · Full text
Structure-Based Discovery of Potent CARM1 Inhibitors for Solid Tumor and Cancer Immunology Therapy
Zhuqing Zhang, Zuhao Guo, Xiaowei Xu et al. · Journal of Medicinal Chemistry · 2021 · 36 citations · Full text
Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor
Jianping Hu, Ying-Qing Wang, Yanlian Li et al. · European Journal of Medicinal Chemistry · 2017 · 35 citations · Full text
Medicinal Chemistry, Bioorganic Chemistry, Biochemistry +12
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