Aaron S. Goetz

The Orphan G Protein-coupled Receptor GPR40 Is Activated by Medium and Long Chain Fatty Acids

Celia P. Briscoe, Mohammad Tadayyon, John L. Andrews et al. · Journal of Biological Chemistry · 2003 · 1.1K citations · Full text

Life Sciences, Biochemistry, Pharmacology +17

Discovery of 7-Methyl-5-(1-{[3-(trifluoromethyl)phenyl]acetyl}-2,3-dihydro-1<i>H</i>-indol-5-yl)-7<i>H</i>-pyrrolo[2,3-<i>d</i>]pyrimidin-4-amine (GSK2606414), a Potent and Selective First-in-Class Inhibitor of Protein Kinase R (PKR)-like Endoplasmic Reticulum Kinase (PERK)

Jeffrey M. Axten, Jesús R. Medina, Yanhong Feng et al. · Journal of Medicinal Chemistry · 2012 · 619 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Characterization of a Novel PERK Kinase Inhibitor with Antitumor and Antiangiogenic Activity

Charity Atkins, Qi Liu, Elisabeth A. Minthorn et al. · Cancer Research · 2013 · 429 citations

Medicine, Oncology, Pharmacology +14

Pharmacological regulation of insulin secretion in MIN6 cells through the fatty acid receptor GPR40: identification of agonist and antagonist small molecules

Celia P. Briscoe, Andrew J. Peat, Stephen C. McKeown et al. · British Journal of Pharmacology · 2006 · 400 citations · Full text

Life Sciences, Endocrinology, Pharmacology +17

BMY 7378 is a selective antagonist of the D subtype of α1-adrenoceptors

Aaron S. Goetz, Holly K. King, Stuart D.C. Ward et al. · European Journal of Pharmacology · 1995 · 302 citations

Medicine, Medicinal Chemistry, Pharmacology +11