Serge Halazy

9-(Difluorophosphonoalkyl)guanines as a new class of multisubstrate analog inhibitors of purine nucleoside phosphorylase

Serge Halazy, Anne Ehrhard, Charles Danzin · Journal of the American Chemical Society · 1991 · 131 citations

Life Sciences, Medicinal Chemistry, Pharmacology +10

Design and Synthesis of the First Generation of Novel Potent, Selective, and in Vivo Active (Benzothiazol-2-yl)acetonitrile Inhibitors of the c-Jun N-Terminal Kinase

P. Gaillard, Isabelle Jeanclaude-Etter, Vittoria Ardissone et al. · Journal of Medicinal Chemistry · 2005 · 126 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

In vitro and in vivo pharmacological profile of AS057278, a selective d-amino acid oxidase inhibitor with potential anti-psychotic properties

Tiziana Adage, Anne‐Cécile Trillat, Anna Quattropani et al. · European Neuropsychopharmacology · 2007 · 117 citations

Medicine, Medicinal Chemistry, Pharmacology +11

Ortho- and para-(difluoromethyl)aryl-β-d-glucosides: A new class of enzyme-activated irreversible inhibitors of β-glucosidases

Serge Halazy, Véronique Berges, Anne Ehrhard et al. · Bioorganic Chemistry · 1990 · 82 citations

Life Sciences, Biochemistry, Medicinal Chemistry +12

Design, Synthesis, and Biological Activity of Novel, Potent, and Selective (Benzoylaminomethyl)thiophene Sulfonamide Inhibitors of c-Jun-N-Terminal Kinase

Thomas Rückle, Marco A. Biamonte, Tania Grippi-Vallotton et al. · Journal of Medicinal Chemistry · 2004 · 62 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13