Patrick Boissin

Metabotropic Glutamate Receptor 5 Negative Allosteric Modulators: Discovery of 2-Chloro-4-[1-(4-fluorophenyl)-2,5-dimethyl-1<i>H</i>-imidazol-4-ylethynyl]pyridine (Basimglurant, RO4917523), a Promising Novel Medicine for Psychiatric Diseases

Georg Jaeschke, Sabine Kolczewski, Will Spooren et al. · Journal of Medicinal Chemistry · 2015 · 63 citations · Full text

Psychotropic Medication, Psychopharmacology, Pharmacotherapy +19

Metabolite Identification via LC‐SPE‐NMR‐MS of the In vitro Biooxidation Products of a Lead mGlu5 Allosteric Antagonist and Impact on the Improvement of Metabolic Stability in the Series

Simona Ceccarelli, Götz Schlotterbeck, Patrick Boissin et al. · ChemMedChem · 2007 · 22 citations

Lead Compounds, Metabolomic Profiling, Lead Identification +18

First total synthesis of (−)-α-conidendrin

Patrick Boissin, Robert Dhal, Eric Brown · Tetrahedron Letters · 1989 · 15 citations

Pharmacology, Organic Chemistry, Synthetic Chemistry +1