Nicole Blaquière

Ruthenium-Catalyzed Dehydrogenation of Ammonia Boranes

Nicole Blaquière, Sarah Diallo-Garcia, Serge I. Gorelsky et al. · Journal of the American Chemical Society · 2008 · 302 citations

Chemical Engineering, Novel Organocatalysts, Engineering +11

Discovery of 2-{3-[2-(1-Isopropyl-3-methyl-1<i>H</i>-1,2–4-triazol-5-yl)-5,6-dihydrobenzo[f]imidazo[1,2-<i>d</i>][1,4]oxazepin-9-yl]-1<i>H</i>-pyrazol-1-yl}-2-methylpropanamide (GDC-0032): A β-Sparing Phosphoinositide 3-Kinase Inhibitor with High Unbound Exposure and Robust in Vivo Antitumor Activity

Chudi Ndubaku, Timothy P. Heffron, Steven T. Staben et al. · Journal of Medicinal Chemistry · 2013 · 174 citations · Full text

Drug Target, Unbound Drug Exposure, Pharmacotherapy +21

Antibody-Mediated Delivery of Chimeric BRD4 Degraders. Part 1: Exploration of Antibody Linker, Payload Loading, and Payload Molecular Properties

Peter S. Dragovich, Thomas H. Pillow, Robert A. Blake et al. · Journal of Medicinal Chemistry · 2021 · 140 citations

NF-κB inducing kinase is a therapeutic target for systemic lupus erythematosus

Hans D. Brightbill, Eric Suto, Nicole Blaquière et al. · Nature Communications · 2018 · 120 citations · Full text

Rapid Synthesis of 1,3,5-Substituted 1,2,4-Triazoles from Carboxylic Acids, Amidines, and Hydrazines

Georgette M. Castanedo, Pamela S. Seng, Nicole Blaquière et al. · The Journal of Organic Chemistry · 2011 · 108 citations

1,3,5-Trisubstituted 1,2,4-Triazoles, Carboxylic Acids, 1,3,5-Substituted 1,2,4-Triazoles +9