THE CONCISE GUIDE TO PHARMACOLOGY 2021/22: G protein‐coupled receptors

S P H Alexander, Arthur Christopoulos, Anthony P. Davenport, +151

British Journal of Pharmacology

The Concise Guide to PHARMACOLOGY 2023/24: G protein-coupled receptors

S P H Alexander, Arthur Christopoulos, Anthony P. Davenport, +162

British Journal of Pharmacology

Drug TargetPeptide ScienceSystem PharmacologySystems PharmacologyMolecular Pharmacology +14

Heptahelical domain of metabotropic glutamate receptor 5 behaves like rhodopsin-like receptors

Cyril Goudet, Florence Gaven, Julie Kniazeff, +6

Proceedings of the National Academy of Sciences

Rhodopsin-like ReceptorsNeurotransmitterInverse AgonistHeptahelical DomainSynaptic Signaling +14

An allosteric modulator to control endogenous G protein-coupled receptors with light

Silvia Pittolo, Xavier Gómez‐Santacana, Kay Eckelt, +8

Nature Chemical Biology

Photoreceptor CellMolecular PhysiologySignal TransductionBiochemistryG Protein-coupled Receptor +9

Evidence for a single heptahelical domain being turned on upon activation of a dimeric GPCR

Veronika Hlaváčková, Cyril Goudet, Julie Kniazeff, +7

The EMBO Journal

Signal TransductionG Protein-coupled ReceptorNatural SciencesMolecular BiologySingle Heptahelical Domain +4

Asymmetric Functioning of Dimeric Metabotropic Glutamate Receptors Disclosed by Positive Allosteric Modulators

Cyril Goudet, Julie Kniazeff, Veronika Hlaváčková, +6

Journal of Biological Chemistry

Metabotropic Glutamate ReceptorsSynaptic TransmissionNeurotransmitterSynaptic SignalingSocial Sciences +17

d-myo-Inositol 1-phosphate as a surrogate of d-myo-inositol 1,4,5-tris phosphate to monitor G protein-coupled receptor activation

Eric Trinquet, Michel Fink, Hervé Bazin, +16

Analytical Biochemistry

Signal TransductionMolecular PhysiologyBiochemistryG Protein-coupled ReceptorMedicine +7

Electrophysiological and behavioral evidence that modulation of metabotropic glutamate receptor 4 with a new agonist reverses experimental parkinsonism

Corinne Beurrier, S. Lopez, Delphine Révy, +8

The FASEB Journal

NeurotransmitterBehavioral EvidenceNeurotransmissionSynaptic SignalingSocial Sciences +15

Group III metabotropic glutamate receptors inhibit hyperalgesia in animal models of inflammation and neuropathic pain

Cyril Goudet, Eric Chapuy, Abdelkrim Alloui, +3

Pain

Acute PainPain MedicineIi MglursNeuropathic PainMolecular Pain +14

N-{4-Chloro-2-[(1,3-dioxo-1,3-dihydro-2H-isoindol-2-yl)methyl]phenyl}-2-hydroxybenzamide (CPPHA) Acts through a Novel Site as a Positive Allosteric Modulator of Group 1 Metabotropic Glutamate Receptors

Yelin Chen, Cyril Goudet, Jean‐Philippe Pin, +1

Molecular Pharmacology