Roland Neuhaus

Selective covalent targeting of GPX4 using masked nitrile-oxide electrophiles

John K. Eaton, Laura Furst, Richard A. Ruberto et al. · Nature Chemical Biology · 2020 · 445 citations · Full text

Selective Covalent Targeting, Organometallic Electrochemistry, Chemistry +1

Identification and Optimization of the First Highly Selective GLUT1 Inhibitor BAY‐876

Hölger Siebeneicher, Arwed Cleve, Hartmut Rehwinkel et al. · ChemMedChem · 2016 · 262 citations · Full text

Pan-mutant IDH1 inhibitor BAY 1436032 for effective treatment of IDH1 mutant astrocytoma in vivo

Stefan Pusch, Sonja Krausert, Viktoria Fischer et al. · Acta Neuropathologica · 2017 · 174 citations

Tumor Biology, Neuro-oncology, Glioma +10

ZK200775: A phosphonate quinoxalinedione AMPA antagonist for neuroprotection in stroke and trauma

Lechosław Turski, Andreas Huth, Malcolm J. Sheardown et al. · Proceedings of the National Academy of Sciences · 1998 · 167 citations · Full text

Pharmaceutical Science, Bioorganic Chemistry, Cerebrovascular Disease +27

Mechanism-Based Inhibition: Deriving KI and kinact Directly from Time-Dependent IC50 Values

Ben‐Fillippo Krippendorff, Roland Neuhaus, Philip Lienau et al. · SLAS DISCOVERY · 2009 · 154 citations · Full text