Adriana Port

Synthesis and Biological Evaluation of the 1-Arylpyrazole Class of σ₁ Receptor Antagonists: Identification of 4-{2-[5-Methyl-1-(naphthalen-2-yl)-1<i>H</i>-pyrazol-3-yloxy]ethyl}morpholine (S1RA, E-52862)

José Luis Dı́az, Rosa Cuberes, Joana Berrocal et al. · Journal of Medicinal Chemistry · 2012 · 128 citations · Full text

Spacer Lengths, Pharmacotherapy, New Series +18

Synthesis and Structure–Activity Relationship Study of a New Series of Selective σ₁Receptor Ligands for the Treatment of Pain: 4-Aminotriazoles

José Luis Dı́az, Ute Christmann, Ariadna Fernández et al. · Journal of Medicinal Chemistry · 2015 · 42 citations · Full text

4-Aryl-1-oxa-4,9-diazaspiro[5.5]undecane Derivatives as Dual μ-Opioid Receptor Agonists and σ₁ Receptor Antagonists for the Treatment of Pain

Mónica Garcı́a, Marina Virgili, Mónica Alonso et al. · Journal of Medicinal Chemistry · 2019 · 33 citations · Full text

Critical comparison of shake-flask, potentiometric and chromatographic methods for lipophilicity evaluation (log P o/w ) of neutral, acidic, basic, amphoteric, and zwitterionic drugs

Adriana Port, Magda Bordas, Raquel Enrech et al. · European Journal of Pharmaceutical Sciences · 2018 · 30 citations · Full text

Pharmaceutical Science, Biochemistry, Medicine +9

Preparation of enantiomers of 1-(1-naphthyl)-2,2-dimethylpropylamine and their behaviour as chiral solvating agents: study of diastereochemic association by Job's plots and intermolecular NOE measurements

Adriana Port, A. Virgili, A. Alvarez‐Larena et al. · Tetrahedron Asymmetry · 2000 · 27 citations

Organic Chemistry, Diastereochemic Association, Stereoselective Synthesis +5