Concepedia
Statistics
Publications
9
Citations
904
H-Index
Active since
2012
Affiliations
TU Dortmund University(Current)
Max Planck Institute of Molecular Physiology
Ruhr University Bochum
German Cancer Research Center
University of Münster
Rajesh Gontla is an author at TU Dortmund University specializing in natural sciences, medicine, and medicinal chemistry.
Top concepts
Natural SciencesMedicineChemistryPharmacologyDrug DiscoveryOrganic ChemistryMedicinal ChemistryBiochemistryChemical BiologyMolecular Biology
Publications per year
2012–2024
General Enantioselective C−H Activation with Efficiently Tunable Cyclopentadienyl Ligands
Zhi‐Jun Jia, Christian Merten, Rajesh Gontla et al. · Angewandte Chemie International Edition · 2017 · 325 citations
Enantioselective Formal C(sp<sup>3</sup>)−H Bond Activation in the Synthesis of Bioactive Spiropyrazolone Derivatives
Houhua Li, Rajesh Gontla, Jana Flegel et al. · Angewandte Chemie International Edition · 2018 · 126 citations
Zhi‐Jun Jia, Christian Merten, Rajesh Gontla et al. · Angewandte Chemie · 2017 · 118 citations
Modular Nature, Asymmetric Catalysis, C−h Activation Reactions +10
Covalent‐Allosteric Kinase Inhibitors
Jörn Weisner, Rajesh Gontla, Leandi Van Der Westhuizen et al. · Angewandte Chemie International Edition · 2015 · 112 citations
Molecular Docking, Molecular Pharmacology, Medicinal Chemistry +15
Preclinical Efficacy of Covalent-Allosteric AKT Inhibitor Borussertib in Combination with Trametinib in <i>KRAS</i>-Mutant Pancreatic and Colorectal Cancer
Jörn Weisner, Ina Landel, Christoph Reintjes et al. · Cancer Research · 2019 · 88 citations
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