Karol Al Ayed

Structure-Based Design of β1i or β5i Specific Inhibitors of Human Immunoproteasomes

Gerjan de Bruin, E.M. Huber, Bo‐Tao Xin et al. · Journal of Medicinal Chemistry · 2014 · 97 citations · Full text

Proteasome Inhibitors, Drug Target, Human Immunoproteasomes +23

Synthetic studies with the brevicidine and laterocidine lipopeptide antibiotics including analogues with enhanced properties and <i>in vivo</i> efficacy

Karol Al Ayed, Ross D. Ballantine, Michael Hoekstra et al. · Chemical Science · 2022 · 29 citations · Full text

Linearization of the Brevicidine and Laterocidine Lipopeptides Yields Analogues That Retain Full Antibacterial Activity

Ross D. Ballantine, Karol Al Ayed, Samantha J. Bann et al. · Journal of Medicinal Chemistry · 2023 · 17 citations · Full text

Bioorganic Chemistry, Peptide Engineering, Antibacterial Activity +19

Structure–Activity Relationship Studies of α-Ketoamides as Inhibitors of the Phospholipase A and Acyltransferase Enzyme Family

Juan Zhou, Elliot D. Mock, Karol Al Ayed et al. · Journal of Medicinal Chemistry · 2020 · 16 citations · Full text

Synthesis and structure–activity relationship studies of N-terminal analogues of the lipopeptide antibiotics brevicidine and laterocidine

Ross D. Ballantine, Karol Al Ayed, Samantha J. Bann et al. · RSC Medicinal Chemistry · 2022 · 14 citations · Full text