Guillermo A. Morales

Dual-activity PI3K–BRD4 inhibitor for the orthogonal inhibition of MYC to block tumor growth and metastasis

Forest H. Andrews, Alok R. Singh, Shweta Joshi et al. · Proceedings of the National Academy of Sciences · 2017 · 119 citations · Full text

Solid-Phase Synthesis of Benzopiperazinones

Guillermo A. Morales, Jeffrey W. Corbett, William F. DeGrado · The Journal of Organic Chemistry · 1998 · 88 citations

4-Aminopiperidine-4-carboxylic Acid:  A Cyclic α,α-Disubstituted Amino Acid for Preparation of Water-Soluble Highly Helical Peptides

Christopher L. Wysong, T. Scott Yokum, Guillermo A. Morales et al. · The Journal of Organic Chemistry · 1996 · 72 citations

Peptide Engineering, Altmetric Attention Score, Organic Chemistry +16

Single Agent and Synergistic Activity of the “First-in-Class” Dual PI3K/BRD4 Inhibitor SF1126 with Sorafenib in Hepatocellular Carcinoma

Alok R. Singh, Shweta Joshi, Adam M. Burgoyne et al. · Molecular Cancer Therapeutics · 2016 · 56 citations · Full text

Synthesis and Cancer Stem Cell-Based Activity of Substituted 5-Morpholino-7<i>H</i>-thieno[3,2-<i>b</i>]pyran-7-ones Designed as Next Generation PI3K Inhibitors

Guillermo A. Morales, Joseph R. Garlich, Jingdong Su et al. · Journal of Medicinal Chemistry · 2013 · 52 citations · Full text

Pharmaceutical Chemistry, Tumor Biology, Medicinal Chemistry +16