Concepedia
Statistics
Publications
8
Citations
205
H-Index
Active since
2004
Affiliations
Cancer Center of Hawaii(Current)
University of Hawaiʻi at Mānoa
University of Hawaii System
University of Hawaii Cancer Center
Cedars-Sinai Medical Center
Francisco Lopez‐Tapia is an author at Cancer Center of Hawaii specializing in medicinal chemistry, natural sciences, and drug discovery.
Top concepts
MedicineBiochemistryPharmacologyDrug DiscoveryDrug DevelopmentNatural SciencesMedicinal ChemistryDrug DesignPharmacotherapyChemical Biology
Publications per year
2004–2022
Hydroxamic Acid and Benzoic Acid–Based STAT3 Inhibitors Suppress Human Glioma and Breast Cancer Phenotypes <i>In Vitro</i> and <i>In Vivo</i>
Peibin Yue, Francisco Lopez‐Tapia, David Paladino et al. · Cancer Research · 2015 · 73 citations · Full text
Discovery of Novel Azetidine Amides as Potent Small-Molecule STAT3 Inhibitors
Christine Brotherton‐Pleiss, Peibin Yue, Yinsong Zhu et al. · Journal of Medicinal Chemistry · 2020 · 34 citations · Full text
Novel Series of Dihydropyridinone P2X7 Receptor Antagonists
Francisco Lopez‐Tapia, Keith A. M. Walker, Christine Brotherton‐Pleiss et al. · Journal of Medicinal Chemistry · 2015 · 26 citations · Full text
Pharmacotherapy, Pharmaceutical Chemistry, Pre-clinical Pharmacology +18
Novel potent azetidine-based compounds irreversibly inhibit Stat3 activation and induce antitumor response against human breast tumor growth in vivo
Peibin Yue, Yinsong Zhu, Christine Brotherton‐Pleiss et al. · Cancer Letters · 2022 · 18 citations · Full text
Linker Variation and Structure–Activity Relationship Analyses of Carboxylic Acid-based Small Molecule STAT3 Inhibitors
Francisco Lopez‐Tapia, Christine Brotherton‐Pleiss, Peibin Yue et al. · ACS Medicinal Chemistry Letters · 2018 · 17 citations · Full text
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