Roberto Carrasco Gomez

Extending the Structure–Activity Relationship of Anthranilic Acid Derivatives As Farnesoid X Receptor Modulators: Development of a Highly Potent Partial Farnesoid X Receptor Agonist

Daniel Merk, Christina Lamers, Khalil Ali Ahmad et al. · Journal of Medicinal Chemistry · 2014 · 53 citations · Full text

Structure–activity Relationship, Drug Target, Glucose Homeostasis +22

Anthranilic acid derivatives as novel ligands for farnesoid X receptor (FXR)

Daniel Merk, Matthias Gabler, Roberto Carrasco Gomez et al. · Bioorganic & Medicinal Chemistry · 2014 · 33 citations · Full text

Biochemistry, Natural Sciences, Medicine +8

Fragmentation of GW4064 led to a highly potent partial farnesoid X receptor agonist with improved drug-like properties

Daniel Flesch, Matthias Gabler, Andreas Lill et al. · Bioorganic & Medicinal Chemistry · 2015 · 17 citations · Full text

Molecular Pharmacology, Biochemistry, G Protein-coupled Receptor +8

Identification of pirinixic acid derivatives bearing a 2-aminothiazole moiety combines dual PPARα/γ activation and dual 5-LO/mPGES-1 inhibition

Thomas Hanke, Christina Lamers, Roberto Carrasco Gomez et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 12 citations · Full text

Molecular Pharmacology, Medicinal Chemistry, Pharmaceutical Chemistry +13