Luca Gentilucci

Endomorphin-1 Analogues Containing β-Proline Are μ-Opioid Receptor Agonists and Display Enhanced Enzymatic Hydrolysis Resistance

Giuliana Cardillo, Luca Gentilucci, Ahmed R. Qasem et al. · Journal of Medicinal Chemistry · 2002 · 104 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

A Straightforward Method for the Synthesis of Alkylidene and Arylidene Malonates Through Proline-Catalyzed Knoevenagel Condensation

Giuliana Cardillo, Serena Fabbroni, Luca Gentilucci et al. · Synthetic Communications · 2003 · 90 citations

Natural Sciences, Chemistry, Catalysis +10

Convenient synthesis of optically active 2H-azirine-2-carboxylic esters by Swern oxidation of aziridine-2-carboxylic esters

Luca Gentilucci, Yvonne Grijzen, L. Thijs et al. · Tetrahedron Letters · 1995 · 79 citations

Natural Sciences, Chemistry, Medicinal Chemistry +9

Synthesis and binding activity of endomorphin-1 analogues containing β-amino acids

Giuliana Cardillo, Luca Gentilucci, Paolo Melchiorre et al. · Bioorganic & Medicinal Chemistry Letters · 2000 · 65 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

Synthesis of enantiomerically pure trans aziridine-2-carboxylates by diastereoselective Gabriel-cromwell reaction

Giuliana Cardillo, Luca Gentilucci, Claudia Tomasini et al. · Tetrahedron Asymmetry · 1996 · 54 citations

Natural Sciences, Chemistry, Medicinal Chemistry +10