Nikolaos Papaioannou

Kinetic Resolution of Alcohols Catalyzed by Tripeptides Containing the <i>N</i>-Alkylimidazole Substructure

Scott J. Miller, Gregory T. Copeland, Nikolaos Papaioannou et al. · Journal of the American Chemical Society · 1998 · 239 citations

Combinatorial Chemistry, Bioorganic Chemistry, Engineering +13

A Biomimetic Approach to Asymmetric Acyl Transfer Catalysis

Elizabeth R. Jarvo, Gregory T. Copeland, Nikolaos Papaioannou et al. · Journal of the American Chemical Society · 1999 · 220 citations

Engineering, Peptide Engineering, Biomimetic Approach +17

Discovery of Clinical Candidate 1-{[(2 <i>S</i> ,3 <i>S</i> ,4 <i>S</i> )-3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin-1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design

Katherine L. Lee, Catherine M. Ambler, David R. Anderson et al. · Journal of Medicinal Chemistry · 2017 · 138 citations · Full text

Enantioselective Synthesis of an Aziridinomitosane and Selective Functionalizations of a Key Intermediate

Nikolaos Papaioannou, Jarred T. Blank, Scott J. Miller · The Journal of Organic Chemistry · 2003 · 40 citations

Enantioselective Synthesis of a Mitosane Core Assisted by Diversity-Based Catalyst Discovery

Nikolaos Papaioannou, Catherine A. Evans, Jarred T. Blank et al. · Organic Letters · 2001 · 33 citations

Bioorganic Chemistry, Engineering, Mitosane 1 +20