Jacob Krall

Design, Synthesis, and Pharmacological Characterization of<i>N</i>- and<i>O</i>-Substituted 5,6,7,8-Tetrahydro-4<i>H</i>-isoxazolo[4,5-<i>d</i>]azepin-3-ol Analogues: Novel 5-HT_2A/5-HT_2CReceptor Agonists with Pro-Cognitive Properties

Anders A. Jensen, Niels Plath, Martin Holst Friborg Pedersen et al. · Journal of Medicinal Chemistry · 2013 · 63 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +15

4-Hydroxy-1,2,3-triazole moiety as bioisostere of the carboxylic acid function: a novel scaffold to probe the orthosteric γ-aminobutyric acid receptor binding site

Alessandro Giraudo, Jacob Krall, Birgitte Nielsen et al. · European Journal of Medicinal Chemistry · 2018 · 32 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Probing α₄βδ GABA_AReceptor Heterogeneity: Differential Regional Effects of a Functionally Selective α₄β₁δ/α₄β₃δ Receptor Agonist on Tonic and Phasic Inhibition in Rat Brain

Kirsten Hoestgaard-Jensen, Nils Ole Dalby, Jacob Krall et al. · Journal of Neuroscience · 2014 · 25 citations · Full text

Medicine, Neuroscience, Pharmacology +16

Novel 4-(Piperidin-4-yl)-1-hydroxypyrazoles as γ-Aminobutyric Acid_A Receptor Ligands: Synthesis, Pharmacology, and Structure−Activity Relationships

Henriette A. Møller, Tommy Sander, Jesper L. Kristensen et al. · Journal of Medicinal Chemistry · 2010 · 24 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Five-Membered <i>N</i>-Heterocyclic Scaffolds as Novel Amino Bioisosteres at γ-Aminobutyric Acid (GABA) Type A Receptors and GABA Transporters

Alessandro Giraudo, Jacob Krall, Francesco Bavo et al. · Journal of Medicinal Chemistry · 2019 · 24 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17