Danial Beaudry

Magnesium Ethoxide Promoted Conversion of Nitriles to Amidines and Its Application in 5,6-Dihydroimidazobenzoxazepine Synthesis

Michael E. Dalziel, Julie A. Deichert, Diane E. Carrera et al. · Organic Letters · 2018 · 21 citations

Pharmacy, Chemistry, Medicinal Chemistry +11

Development of an Efficient Manufacturing Process for Reversible Bruton’s Tyrosine Kinase Inhibitor GDC-0853

Haiming Zhang, Theresa Cravillion, Ngiap‐Kie Lim et al. · Organic Process Research & Development · 2018 · 18 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Manufacture of the PI3K β-Sparing Inhibitor Taselisib. Part 2: Development of a Highly Efficient and Regioselective Late-Stage Process

Frédéric St-Jean, Travis Remarchuk, Rémy Angelaud et al. · Organic Process Research & Development · 2019 · 16 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Improved Synthesis of the Nav1.7 Inhibitor GDC-0276 via a Highly Regioselective S_NAr Reaction

Andreas Stumpf, Zhigang Ken Cheng, Danial Beaudry et al. · Organic Process Research & Development · 2019 · 16 citations

Pharmacy, Chemistry, Medicinal Chemistry +10

Development of a Practical and Greener Process for the Dual Leucine Zipper Kinase Inhibitor GDC-0134 Comprising Two S_NAr Reactions, Oxidation and Suzuki Coupling

Fabienne Hoffmann-Emery, Katrin Niedermann, Pankaj D. Rege et al. · Organic Process Research & Development · 2022 · 14 citations

Pharmacy, Chemical Engineering, Chemistry +12