Petra Johannesson

Vinyl Sulfide Cyclized Analogues of Angiotensin II with High Affinity and Full Agonist Activity at the AT₁Receptor

Petra Johannesson, Gunnar Lindeberg, Anja Johansson et al. · Journal of Medicinal Chemistry · 2002 · 122 citations · Full text

Organic Chemistry, Peptide Science, Pharmacotherapy +18

Discovery of Second Generation Reversible Covalent DPP1 Inhibitors Leading to an Oxazepane Amidoacetonitrile Based Clinical Candidate (AZD7986)

Kevin Doyle, Hans Lönn, Helena Käck et al. · Journal of Medicinal Chemistry · 2016 · 80 citations · Full text

Drug Target, Clinical Candidate, Pharmacotherapy +19

Involvement of the metabolic sensor GPR81 in cardiovascular control

Kristina Wallenius, Pia Thalén, Jan‐Arne Björkman et al. · JCI Insight · 2017 · 57 citations · Full text

Hypertension, Metabolic Remodeling, Gpr81 Agonism +19

Synthesis and Functionalization of Cyclic Sulfonimidamides: A Novel Chiral Heterocyclic Carboxylic Acid Bioisostere

Nils Pemberton, Henrik Gradén, Emma Evertsson et al. · ACS Medicinal Chemistry Letters · 2012 · 55 citations · Full text

Bioorganic Chemistry, Engineering, Amino Acid +14

Design and Optimization of Pyrazinecarboxamide-Based Inhibitors of Diacylglycerol Acyltransferase 1 (DGAT1) Leading to a Clinical Candidate Dimethylpyrazinecarboxamide Phenylcyclohexylacetic Acid (AZD7687)

Jonas G. Barlind, Udo Bauer, Alan M. Birch et al. · Journal of Medicinal Chemistry · 2012 · 36 citations · Full text

Pharmaceutical Science, Candidate Drug, Pyrazinecarboxamide Dgat1 Inhibitors +17