Reversal of tumoral immune resistance by inhibition of tryptophan 2,3-dioxygenase

Luc Pilotte, Pierre Larrieu, Vincent Stroobant, +8

Proceedings of the National Academy of Sciences

ImmunotoxicologyImmunologyImmunoeditingCell DeathImmunotherapy +16

Tryptophan 2,3-Dioxygenase (TDO) Inhibitors. 3-(2-(Pyridyl)ethenyl)indoles as Potential Anticancer Immunomodulators

Eduard Dolušić, Pierre Larrieu, Laurence Moineaux, +8

Journal of Medicinal Chemistry

ImmunologyTryptophan DegradationCell DeathPharmaceutical ChemistryMolecular Pharmacology +17

Efficient synthesis of aryldipyrromethanes in water and their application in the synthesis of corroles and dipyrromethenes

Taoufik Rohand, Eduard Dolušić, Thien H. Ngo, +2

ARKIVOC

Gold Electrode Incorporating Corrole as an Ion-Channel Mimetic Sensor for Determination of Dopamine

Katarzyna Kurzątkowska, Eduard Dolušić, Wim Dehaen, +3

Analytical Chemistry

Discovery and preliminary SARs of keto-indoles as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

Eduard Dolušić, Pierre Larrieu, Sébastien Blanc, +15

European Journal of Medicinal Chemistry

Medicinal ChemistryBiochemistryPreliminary SarsNatural SciencesMedicine +4

Synthesis, evaluation and structure-activity relationship of new 3-carboxamide coumarins as FXIIa inhibitors

Charlotte Bouckaert, Silvia Serra, G. Rondelet, +5

European Journal of Medicinal Chemistry

Fxiia InhibitorsMedicinal ChemistryNew 3-Carboxamide CoumarinsPharmaceutical ScienceBiochemistry +9

Indol-2-yl ethanones as novel indoleamine 2,3-dioxygenase (IDO) inhibitors

Eduard Dolušić, Pierre Larrieu, Sébastien Blanc, +15

Bioorganic & Medicinal Chemistry

Medicinal ChemistryBiochemistryMedicineNatural SciencesIndol-2-yl Ethanones +3

Indoleamine 2,3-dioxygenase inhibitory activity of derivatives of marine alkaloid tsitsikammamine A

Eduard Dolušić, Pierre Larrieu, Céline Meinguet, +11

Bioorganic & Medicinal Chemistry Letters

Aldehyde DehydrogenaseBiochemistryNatural SciencesSecondary MetaboliteChemical Biology +1

Porphotetramethenes with 1,3-alternate conformation of pyrrole rings from oxidative N-alkylation of porphyrin tetraphenols

Eduard Dolušić, Suzanne Toppet, S. Smeets, +3

Tetrahedron

Combinatorial ChemistryChemical EngineeringEngineeringPyrrole RingsOrganic Chemistry +4

Biotinylated Indoles as Probes for Indole-Binding Proteins

Eduard Dolušić, Mariusz Kowalczyk, Volker Magnus, +2

Bioconjugate Chemistry