Concepedia

T.B. Shaik

TS

Statistics

Publications

10

Citations

617

H-Index

10

Active since

2016

Affiliations

Centre National de la Recherche Scientifique(Current)

University of Freiburg

Institut de génétique et de biologie moléculaire et cellulaire

Inserm

Université de Strasbourg

T.B. Shaik is an author at Centre National de la Recherche Scientifique specializing in drug discovery, enzyme inhibition, and medicinal chemistry.

ORCID

Publications per year

2016–2021

10

Publications

10

Structure-Based Design and Synthesis of Novel Inhibitors Targeting HDAC8 from <i>Schistosoma mansoni</i> for the Treatment of Schistosomiasis

Tino Heimburg, Alokta Chakrabarti, Julien Lancelot et al. · Journal of Medicinal Chemistry · 2016 · 123 citations · Full text

, , +17

Characterization of Histone Deacetylase 8 (HDAC8) Selective Inhibition Reveals Specific Active Site Structural and Functional Determinants

Martin Marek, T.B. Shaik, Tino Heimburg et al. · Journal of Medicinal Chemistry · 2018 · 118 citations · Full text

, , +15

Synthesis and Biological Investigation of Phenothiazine-Based Benzhydroxamic Acids as Selective Histone Deacetylase 6 Inhibitors

Katharina Vögerl, Nghia Ong, Johanna Senger et al. · Journal of Medicinal Chemistry · 2019 · 101 citations · Full text

, , +17

Structure-Based Design and Biological Characterization of Selective Histone Deacetylase 8 (HDAC8) Inhibitors with Anti-Neuroblastoma Activity

Tino Heimburg, Fiona R. Kolbinger, Patrik Zeyen et al. · Journal of Medicinal Chemistry · 2017 · 93 citations · Full text

, , +16

Novel spiroindoline HDAC inhibitors: Synthesis, molecular modelling and biological studies

Margherita Brindisi, Johanna Senger, Caterina Cavella et al. · European Journal of Medicinal Chemistry · 2018 · 50 citations · Full text

, , +13

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