Laure Dufau

Dimerized Linear Mimics of a Natural Cyclopeptide (TMC-95A) Are Potent Noncovalent Inhibitors of the Eukaryotic 20S Proteasome

Audrey Desvergne, Emilie Génin, Xavier Maréchal et al. · Journal of Medicinal Chemistry · 2013 · 38 citations · Full text

Pharmacy, Biochemistry, Medicinal Chemistry +17

Dimer Disruption and Monomer Sequestration by Alkyl Tripeptides Are Successful Strategies for Inhibiting Wild-Type and Multidrug-Resistant Mutated HIV-1 Proteases

Ludovic Bannwarth, Thierry Rose, Laure Dufau et al. · Biochemistry · 2008 · 26 citations

Life Sciences, Biochemistry, Molecular Biology +15

α- and β-hydrazino acid-based pseudopeptides inhibit the chymotrypsin-like activity of the eukaryotic 20S proteasome

Andrea Bordessa, Massaba Keita, Xavier Maréchal et al. · European Journal of Medicinal Chemistry · 2013 · 21 citations

Life Sciences, Biochemistry, Medicinal Chemistry +12

Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild‐Type and Mutated HIV‐1 Protease Dimerization

Anamaria Vidu, Laure Dufau, Ludovic Bannwarth et al. · ChemMedChem · 2010 · 19 citations

Pharmacy, Biochemistry, Medicinal Chemistry +16

New C4- and C1-derivatives of furo[3,4-c]pyridine-3-ones and related compounds: Evidence for site-specific inhibition of the constitutive proteasome and its immunoisoform

Anna Hovhannisyan, The Hien Pham, Dominique Bouvier et al. · Bioorganic & Medicinal Chemistry Letters · 2014 · 19 citations · Full text

Life Sciences, Biochemistry, Chemistry +11