Valerio Gatti

Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at Indole-2-carboxamide

Giuseppe La Regina, Antonio Coluccia, Andrea Brancale et al. · Journal of Medicinal Chemistry · 2011 · 160 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Computer-aided identification, design and synthesis of a novel series of compounds with selective antiviral activity against chikungunya virus

Marcella Bassetto, Tine De Burghgraeve, Leen Delang et al. · Antiviral Research · 2013 · 106 citations · Full text

Pharmacy, Infectious Diseases, Medicinal Chemistry +10

New Arylthioindoles and Related Bioisosteres at the Sulfur Bridging Group. 4. Synthesis, Tubulin Polymerization, Cell Growth Inhibition, and Molecular Modeling Studies

Giuseppe La Regina, Taradas Sarkar, Ruoli Bai et al. · Journal of Medicinal Chemistry · 2009 · 88 citations · Full text

Pharmacy, Biochemistry, Medicinal Chemistry +15

Design and Synthesis of 2-Heterocyclyl-3-arylthio-1<i>H</i>-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability

Giuseppe La Regina, Ruoli Bai, Willeke Rensen et al. · Journal of Medicinal Chemistry · 2011 · 75 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Synthesis, structure–activity relationships and molecular modeling studies of new indole inhibitors of monoamine oxidases A and B

Giuseppe La Regina, Romano Silvestri, Valerio Gatti et al. · Bioorganic & Medicinal Chemistry · 2008 · 33 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16