Yoshihiro Sugihara

Electroorganic chemistry. 60. Electroorganic synthesis of enamides and enecarbamates and their utilization in organic synthesis

Tatsuya Shono, Yoshihiro Matsumura, Kenji Tsubata et al. · Journal of the American Chemical Society · 1982 · 206 citations

Electroorganic Synthesis, Bioorganic Chemistry, Engineering +12

Discovery of a Piperidine-4-carboxamide CCR5 Antagonist (TAK-220) with Highly Potent Anti-HIV-1 Activity

Shinichi Imamura, Takashi Ichikawa, Youichi Nishikawa et al. · Journal of Medicinal Chemistry · 2006 · 71 citations · Full text

Highly Potent Inhibition of Human Immunodeficiency Virus Type 1 Replication by TAK-220, an Orally Bioavailable Small-Molecule CCR5 Antagonist

Katsunori Takashima, Hiroshi Miyake, Naoyuki Kanzaki et al. · Antimicrobial Agents and Chemotherapy · 2005 · 59 citations · Full text

Medicine, Human Retrovirus, Highly Potent Inhibition +14

CCR5 antagonists as anti-HIV-1 agents. Part 3: Synthesis and biological evaluation of piperidine-4-carboxamide derivatives

Shinichi Imamura, Youichi Nishikawa, Takashi Ichikawa et al. · Bioorganic & Medicinal Chemistry · 2004 · 45 citations

Piperidine-4-carboxamide Derivatives, Medicine, Immunology +10

CCR5 Antagonists as Anti-HIV-1 Agents. 1. Synthesis and Biological Evaluation of 5-Oxopyrrolidine-3-carboxamide Derivatives

Shinichi Imamura, Yuji Ishihara, Taeko Hattori et al. · Chemical and Pharmaceutical Bulletin · 2004 · 37 citations · Full text