Ciro J. Spagnuolo

An integrated approach to the selection of optimal salt form for a new drug candidate

Kenneth R. Morris, M. Fakes, Ajit B. Thakur et al. · International Journal of Pharmaceutics · 1994 · 146 citations

Medicinal Chemistry, Integrated Approach, Pharmaceutical Science +11

Synthesis and antimuscarinic properties of some N-substituted 5-(aminomethyl)-3,3-diphenyl-2(3H)-furanones

Carl Kaiser, Ciro J. Spagnuolo, Theodore C. Adams et al. · Journal of Medicinal Chemistry · 1992 · 33 citations

Medicinal Chemistry, Antimuscarinic Properties, Heterocyclic +14

Analogs of oxybutynin. Synthesis and antimuscarinic and bladder activity of some substituted 7-amino-1-hydroxy-5-heptyn-2-ones and related compounds

J. Paul Carter, Lalita Noronha‐Blob, Vicki H. Audia et al. · Journal of Medicinal Chemistry · 1991 · 28 citations

γ-alkylation of α,β-unsaturated ketones: α'-phenylsulfonyl groups as regioselective control elements

Peter T. Lansbury, Gregory E. Bebernitz, Susan C. Maynard et al. · Tetrahedron Letters · 1985 · 24 citations

Engineering, Regioselective Control Elements, Organic Chemistry +5

Trifluoroacetic Acid-Mediated Cleavage of a Triethylsilyl Protecting Group:  Application in the Final Step of the Semisynthetic Route to Paclitaxel (Taxol)

Ambarish K. Singh, Raymond E. Weaver, Gerald L. Powers et al. · Organic Process Research & Development · 2002 · 19 citations

Aqueous Acetic Acid, Pharmaceutical Science, Bioorganic Chemistry +17