Orally Active and Potent Inhibitors of γ-Aminobutyric Acid Uptake

Fadia E. Ali, William E. Bondinell, Penelope A. Dandridge, +15

Journal of Medicinal Chemistry

PharmacotherapyExperimental PharmacologyMolecular PharmacologyMedicinal ChemistryGaba Uptake +14

Absolute stereochemistry and dopaminergic activity of enantiomers of 2,3,4,5-tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine

Carl Kaiser, Penelope A. Dandridge, Eleanor Garvey, +5

Journal of Medicinal Chemistry

Organic ChemistryPharmacotherapyR IsomerPharmaceutical ChemistryMedicinal Chemistry +14

Studies on renal dopamine receptors with a new agonist

Robert G. Pendleton, Lucinda Samler, Carl Kaiser, +1

European Journal of Pharmacology

Functional SelectivityMedicineRenal Dopamine ReceptorsDopaminePharmacology +1

2-Substituted Cyclopropylamines. II. Effect of Structure upon Monoamine Oxidase-Inhibitory Activity as Measured <i>in Vivo</i> by Potentiation of Tryptamine Convulsions

Charles L. Zirkle, Carl Kaiser, David H. Tedeschi, +2

Journal of Medicinal Chemistry

2-Substituted CyclopropylaminesNeurotransmitterAltmetric Attention ScorePharmacotherapyChemical Biology +18

Preparation of Some Cyclopropanes and Stable Sulfoxonium Ylides from Dimethylsulfoxonium Methylide

Carl Kaiser, Barry M. Trost, James G. Beeson, +1

The Journal of Organic Chemistry

Chemical EngineeringMolecular SciencesEngineeringHeterocyclicChemical Measurement +13

Synthesis, resolution, absolute stereochemistry, and enantioselectivity of 3',4'-dihydroxynomifensine

Penelope A. Dandridge, Carl Kaiser, Martin Brenner, +5

Journal of Medicinal Chemistry

Organic ChemistryDopamine ReceptorsPharmacotherapyChemistryExperimental Pharmacology +17

Some benzyl-substituted imidazoles, triazoles, tetrazoles, pyridinethiones, and structural relatives as multisubstrate inhibitors of dopamine .beta.-hydroxylase. 4. Structure-activity relationships at the copper binding site

Lawrence I. Kruse, Carl Kaiser, Walter E. DeWolf, +6

Journal of Medicinal Chemistry

Multisubstrate inhibitors of dopamine .beta.-hydroxylase. 2. Structure-activity relationships at the phenethylamine binding site

Lawrence I. Kruse, Carl Kaiser, Walter E. DeWolf, +6

Journal of Medicinal Chemistry

Drug TargetPharmacotherapyChemical BiologyPharmaceutical ChemistryMedicinal Chemistry +17

2-Substituted Cyclopropylamines. I. Derivatives and Analogs of 2-Phenylcyclopropylamine

Carl Kaiser, Bruce M. Lester, Charles L. Zirkle, +4

Journal of Medicinal Chemistry

Medicinal ChemistryDerivativesHeterocyclicI. DerivativesNatural Sciences +8

Substituted 1-benzylimidazole-2-thiols as potent and orally active inhibitors of dopamine .beta.-hydroxylase

Lawrence I. Kruse, Carl Kaiser, Walter E. DeWolf, +6

Journal of Medicinal Chemistry

Drug TargetAltmetric Attention ScorePharmacotherapyPharmaceutical ChemistryMolecular Pharmacology +16