Bart Harper

(2<i>S</i>,3<i>S</i>)-3-Amino-4-(3,3-difluoropyrrolidin-1-yl)-<i>N,N</i>-dimethyl-4-oxo-2-(4-[1,2,4]triazolo[1,5-<i>a</i>]- pyridin-6-ylphenyl)butanamide:  A Selective α-Amino Amide Dipeptidyl Peptidase IV Inhibitor for the Treatment of Type 2 Diabetes

Scott D. Edmondson, Anthony Mastracchio, Robert J. Mathvink et al. · Journal of Medicinal Chemistry · 2006 · 121 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +16

Discovery of Vibegron: A Potent and Selective β₃Adrenergic Receptor Agonist for the Treatment of Overactive Bladder

Scott D. Edmondson, Cheng Zhu, Nam Fung Kar et al. · Journal of Medicinal Chemistry · 2015 · 102 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

2-Substituted piperazine-derived imidazole carboxamides as potent and selective CCK1R agonists for the treatment of obesity

Richard Berger, Cheng Zhu, Alexa R. Hansen et al. · Bioorganic & Medicinal Chemistry Letters · 2008 · 30 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +11

Discovery of 3-aminopiperidines as potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitors

Jason M. Cox, Bart Harper, Anthony Mastracchio et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +8

Design, Synthesis, and Evaluation of Conformationally Restricted Acetanilides as Potent and Selective β₃Adrenergic Receptor Agonists for the Treatment of Overactive Bladder

Christopher R. Moyes, Richard Berger, Stephen D. Goble et al. · Journal of Medicinal Chemistry · 2014 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15