Concepedia
Statistics
Publications
7
Citations
307
H-Index
Active since
2012
Affiliations
Technische Universität Darmstadt(Current)
Helmholtz Institute for Pharmaceutical Research Saarland
Heiko Fittler is an author at Technische Universität Darmstadt specializing in ligand binding, pharmacy, and drug design.
Publications per year
2012–2016
Combinatorial Optimization of Cystine-Knot Peptides towards High-Affinity Inhibitors of Human Matriptase-1
Bernhard Glotzbach, Michael Reinwarth, Niklas Weber et al. · PLoS ONE · 2013 · 64 citations · Full text
Pharmacy, Biochemistry, Medicinal Chemistry +17
Locked by Design: A Conformationally Constrained Transglutaminase Tag Enables Efficient Site‐Specific Conjugation
Vanessa Siegmund, Stefan Schmelz, Stephan Dickgießer et al. · Angewandte Chemie International Edition · 2015 · 55 citations
Pharmacy, Biochemistry, Molecular Biology +17
Combinatorial tuning of peptidic drug candidates: high-affinity matriptase inhibitors through incremental structure-guided optimization
Heiko Fittler, Olga Avrutina, Bernhard Glotzbach et al. · Organic & Biomolecular Chemistry · 2013 · 51 citations
Pharmacy, Medicinal Chemistry, Pharmacology +17
Potent inhibitors of human matriptase‐1 based on the scaffold of sunflower trypsin inhibitor
Heiko Fittler, Olga Avrutina, Martin Empting et al. · Journal of Peptide Science · 2014 · 46 citations
Pharmacy, Medicinal Chemistry, Pharmacology +16
An Apoptosis‐Inducing Peptidic Heptad That Efficiently Clusters Death Receptor 5
Bernhard Valldorf, Heiko Fittler, Lukas Deweid et al. · Angewandte Chemie International Edition · 2016 · 37 citations
Life Sciences, Molecular Biology, Oncology +17
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