Joel Goldberg

Small-molecule antagonists of Myc/Max dimerization inhibit Myc-induced transformation of chicken embryo fibroblasts

Thorsten Berg, Steven B. Cohen, Joel Desharnais et al. · Proceedings of the National Academy of Sciences · 2002 · 323 citations · Full text

Discovery of Clinical Candidate 1-{[(2 <i>S</i> ,3 <i>S</i> ,4 <i>S</i> )-3-Ethyl-4-fluoro-5-oxopyrrolidin-2-yl]methoxy}-7-methoxyisoquinoline-6-carboxamide (PF-06650833), a Potent, Selective Inhibitor of Interleukin-1 Receptor Associated Kinase 4 (IRAK4), by Fragment-Based Drug Design

Katherine L. Lee, Catherine M. Ambler, David R. Anderson et al. · Journal of Medicinal Chemistry · 2017 · 138 citations · Full text

Two Comparisons of the Performance of Positional Scanning and Deletion Synthesis for the Identification of Active Constituents in Mixture Combinatorial Libraries

Dale L. Boger, Jae Kyoo Lee, Joel Goldberg et al. · The Journal of Organic Chemistry · 2000 · 73 citations

Erythropoietin Mimetics Derived from Solution Phase Combinatorial Libraries

Joel Goldberg, Qing Jin, Yves Ambroise et al. · Journal of the American Chemical Society · 2001 · 67 citations

Biomedical Engineering, Medicinal Chemistry, Receptor Tyrosine Kinase +16

Duocarmycin SA Shortened, Simplified, and Extended Agents:  A Systematic Examination of the Role of the DNA Binding Subunit

Dale L. Boger, Donald L. Hertzog, Bernd Bollinger et al. · Journal of the American Chemical Society · 1997 · 66 citations