Craig S. Harris

Injectable Self-Healing Hydrogels Based on Boronate Ester Formation between Hyaluronic Acid Partners Modified with Benzoxaborin Derivatives and Saccharides

Tamiris Vilas Boas Figueiredo, Jing Jing, Isabelle Jeacomine et al. · Biomacromolecules · 2019 · 109 citations · Full text

Inhibitors of epidermal growth factor receptor tyrosine kinase: Novel C-5 substituted anilinoquinazolines designed to target the ribose pocket

Peter Ballard, Robert H. Bradbury, Craig S. Harris et al. · Bioorganic & Medicinal Chemistry Letters · 2005 · 40 citations · Full text

Medicinal Chemistry, Biochemistry, Medicine +11

Boronic acid and diol-containing polymers: how to choose the correct couple to form “strong” hydrogels at physiological pH

Tamiris Vilas Boas Figueiredo, Vanina A. Cosenza, Yu Ogawa et al. · Soft Matter · 2020 · 40 citations · Full text

Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists

Gilles Ouvry, Claire Bouix‐Peter, Fabrice Ciesielski et al. · Bioorganic & Medicinal Chemistry Letters · 2016 · 37 citations · Full text

Molecular Pharmacology, Drug Target, Medicine +6

Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1,3,4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1,2,4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancers

Bernard Barlaam, Sabina Cosulich, Bénédicte Delouvrié et al. · Bioorganic & Medicinal Chemistry Letters · 2015 · 35 citations

Medicinal Chemistry, Medicine, Selective Inhibitor +9