CrystEngComm · 2023 · 11 citations · 45 references
PharmacyPharmaceuticsPharmacotherapyAntimicrobial PharmacotherapyBioavailabilityDissolution TestingDissolution MediaDrug DissolutionDrug SolubilityFormulation Effects On DissolutionSolubility EnhancementSolubility OptimizationBacteriostatic ActivityBacteriostatic AgentsDissolution OptimizationHigh SolubilityPoorly Water-soluble DrugsSolubilitySolubility DeterminationWater Sorption And Solubility
Trimethoprim (TMP) is a commonly used BCS class II antibiotic, the water solubility of which needs to be improved to overcome the limitations in oral administration.
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A short history of<i>SHELX</i>
George M. Sheldrick · Acta Crystallographica Section A Foundations of Crystallography · 2007 · 87.4K citations · Full text
VMD: Visual molecular dynamics
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