Asymmetric synthesis of pyrrolo[2,3–b]indole scaffolds by organocatalytic [3 + 2] dearomative annulation

Chemistry of the Hexahydropyrrolo[2,3-<i>b</i>]indoles:  Configuration, Conformation, Reactivity, and Applications in Synthesis

David Crich, Abhisek Banerjee · Accounts of Chemical Research · 2007 · 410 citations

Natural Sciences, Chemistry, Medicinal Chemistry +14

Control of Diastereoselectivity in Tandem Asymmetric Reactions Generating Nonadjacent Stereocenters with Bifunctional Catalysis by Cinchona Alkaloids

Baomin Wang, Fanghui Wu, Yi Wang et al. · Journal of the American Chemical Society · 2007 · 360 citations

Pharmacy, Chemistry, Medicinal Chemistry +15

Copper-Catalyzed Highly Enantioselective Cyclopentannulation of Indoles with Donor–Acceptor Cyclopropanes

Xiong Hu, Hao Xu, Saihu Liao et al. · Journal of the American Chemical Society · 2013 · 356 citations

Natural Sciences, Chemistry, Medicinal Chemistry +15

Cupreines and Cupreidines: An Emerging Class of Bifunctional Cinchona Organocatalysts

Tommaso Marcelli, Jan H. van Maarseveen, Henk Hiemstra · Angewandte Chemie International Edition · 2006 · 351 citations

Natural Sciences, Chemistry, Medicinal Chemistry +12

Enantioselective Copper-Catalyzed Construction of Aryl Pyrroloindolines via an Arylation–Cyclization Cascade

Shaolin Zhu, David W. C. MacMillan · Journal of the American Chemical Society · 2012 · 306 citations

Pharmacy, Chemistry, Medicinal Chemistry +15