Concepedia

Development of [<sup>18</sup>F]AmBF<sub>3</sub> Tetrazine for Radiolabeling of Peptides: Preclinical Evaluation and PET Imaging of [<sup>18</sup>F]AmBF<sub>3</sub>-PEG<sub>7</sub>-Tyr<sup>3</sup>-Octreotide in an AR42J Pancreatic Carcinoma Model

Sofia Otaru, Andreas Paulus, Surachet Imlimthan, Iida Kuurne, Helena E. Virtanen, Heidi Liljenbäck, Tuula Tolvanen, Tatsiana Auchynnikava, Anne Roivainen, K. Helariutta,

Bioconjugate Chemistry · 2022 · 20 citations · 24 references

DOIFull text

Open access

Concepts

Abstract

-Tz demonstrated that it offers potential as a prosthetic group for rapid radiolabeling of biomolecules in mild conditions using bioorthogonal chemistry.

References

24

Radiolabeled Peptides: Valuable Tools for the Detection and Treatment of Cancer

Melpomeni Fani, Helmut R. Maëcke, Subhani M. Okarvi · Theranostics · 2012 · 330 citations · Full text

, , +17

Late-stage [<sup>18</sup>F]fluorination: new solutions to old problems

Allen F. Brooks, Joseph J. Topczewski, Naoko Ichiishi et al. · Chemical Science · 2014 · 305 citations · Full text

, , +8

<sup>18</sup>F‐Labeling of Peptides by means of an Organosilicon‐Based Fluoride Acceptor

Ralf Schirrmacher, G. Bradtmoller, Esther Schirrmacher et al. · Angewandte Chemie International Edition · 2006 · 230 citations

, , +14

An Organotrifluoroborate for Broadly Applicable One‐Step <sup>18</sup> F‐Labeling

Zhibo Liu, Maral Pourghiasian, Mark Alex Radtke et al. · Angewandte Chemie International Edition · 2014 · 156 citations

, , +17

Somatostatin receptor PET ligands - the next generation for clinical practice.

Elin Pauwels, Frederik Cleeren, Guy Bormans et al. · PubMed · 2018 · 141 citations · Full text

, , +17