Concepedia

Development of an automated screen for Kv7.2 potassium channels and discovery of a new agonist chemotype

Ciria C. Hernández, Rahilla A. Tarfa, Jose Miguel I. Limcaoco, Ruiting Liu, Pravat Mondal, Clare Hill, Keith Duncan, Thanos Tzounopoulos, Corey R. J. Stephenson, Matthew J. O’Meara,

Bioorganic & Medicinal Chemistry Letters · 2022 · 11 citations · 21 references

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21

RosettaLigand Docking with Full Ligand and Receptor Flexibility

Ian Davis, David Baker · Journal of Molecular Biology · 2008 · 441 citations

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Activation of Expressed KCNQ Potassium Currents and Native Neuronal M-Type Potassium Currents by the Anti-Convulsant Drug Retigabine

L. Tatulian, Patrick Delmas, Fe C. Abogadie et al. · Journal of Neuroscience · 2001 · 404 citations · Full text

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Mediation of Neuronal Apoptosis by Kv2.1-Encoded Potassium Channels

Sumon K. Pal, Karen A. Hartnett, Jeanne M. Nerbonne et al. · Journal of Neuroscience · 2003 · 248 citations · Full text

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Ligand Pose and Orientational Sampling in Molecular Docking

Ryan G. Coleman, Michael Carchia, Teague Sterling et al. · PLoS ONE · 2013 · 225 citations · Full text

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Pathogenic plasticity of Kv7.2/3 channel activity is essential for the induction of tinnitus

Shuang Li, Veronica Choi, Thanos Tzounopoulos · Proceedings of the National Academy of Sciences · 2013 · 163 citations · Full text

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