Concepedia

Fentanyl but not Morphine Interacts with Nonopioid Recombinant Human Neurotransmitter Receptors and Transporters

Randy Torralva, Amy J. Eshleman, Tracy L. Swanson, Jennifer L. Schmachtenberg, William E. Schutzer, Shelley H. Bloom, Katherine M. Wolfrum, John F. Reed, Aaron Janowsky

Journal of Pharmacology and Experimental Therapeutics · 2020 · 71 citations · 63 references

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63

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

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Intravenous fentanyl kinetics

Deborah A. McClain, Carl C. Hug · Clinical Pharmacology & Therapeutics · 1980 · 520 citations

, , +14

Distinct pharmacological properties and distribution in neurons and endocrine cells of two isoforms of the human vesicular monoamine transporter.

Jeffrey D. Erickson, Monika Schäfer, Tom I. Bonner et al. · Proceedings of the National Academy of Sciences · 1996 · 477 citations

, , +16

Modulation by mu-opioid agonists of guanosine-5'-O-(3-[35S]thio)triphosphate binding to membranes from human neuroblastoma SH-SY5Y cells.

John R. Traynor, Stefan R. Nahorski · Molecular Pharmacology · 1995 · 462 citations

, , +17

Drugs Most Frequently Involved in Drug Overdose Deaths: United States, 2011-2016.

Holly Hedegaard, Brigham Bastian, James P. Trinidad et al. · PubMed · 2018 · 402 citations

, , +7