Concepedia
Bioorganic Chemistry · 2019 · 37 citations · 47 references
PharmacyMedicinal ChemistryPharmacologyDrug DesignDrug DiscoveryMolecular PharmacologyLigand BindingProtein BindingPlasma Albumin
47
Crystal structure refinement with<i>SHELXL</i>
George M. Sheldrick · Acta Crystallographica Section C Structural Chemistry · 2014 · 42.5K citations · Full text
Natural Sciences, Chemistry, Computational Chemistry +16
Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
Christopher A. Lipinski, Franco Lombardo, Beryl W. Dominy et al. · Advanced Drug Delivery Reviews · 1997 · 11.2K citations
Pharmacy, Pharmacokinetics, Pharmacology +16
Thermodynamics of protein association reactions: forces contributing to stability
Philip D. Ross, Sankaran Subramanian · Biochemistry · 1981 · 5.5K citations
Natural Sciences, Biochemistry, Biophysics +15
Determination of pKa values of active pharmaceutical ingredients
Sandra Babić, Alka J.M. Horvat, Dragana Mutavdžić Pavlović et al. · TrAC Trends in Analytical Chemistry · 2007 · 501 citations
Pharmacy, Pharmaceutical Analysis, Pharmaceutics +10
Discovery of Alogliptin: A Potent, Selective, Bioavailable, and Efficacious Inhibitor of Dipeptidyl Peptidase IV
Jun Feng, Zhiyuan Zhang, Michael B. Wallace et al. · Journal of Medicinal Chemistry · 2007 · 404 citations · Full text
Medicine, Medicinal Chemistry, Pharmacology +6