Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability

Daniel Silqueira Martins Guimarães, Letícia Silveira de Sousa Luz, Sara Batista do Nascimento, Lorena Rabelo Silva, Natália Rezende de Miranda Martins, Heloísa Gonçalves de Almeida, Vitória de Souza Reis, Sarah El Chamy Maluf, Alexandre Budu, Juliane Aparecida Marinho,

European Journal of Pharmaceutical Sciences · 2019 · 14 citations · 38 references

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