An approach to alicyclic ring-fused xanthines

Escape from Flatland: Increasing Saturation as an Approach to Improving Clinical Success

Frank Lovering, Jack Bikker, Christine Humblet · Journal of Medicinal Chemistry · 2009 · 4.4K citations

Pharmacy, Chemistry, Medicinal Chemistry +8

Property Distributions:  Differences between Drugs, Natural Products, and Molecules from Combinatorial Chemistry

Miklós Fehér, Jonathan M. Schmidt · Journal of Chemical Information and Computer Sciences · 2002 · 921 citations

Pharmacy, Chemistry, Medicinal Chemistry +16

Parallel Synthesis of a Library of Benzoxazoles and Benzothiazoles Using Ligand-Accelerated Copper-Catalyzed Cyclizations of <i>ortho</i>-Halobenzanilides

Ghotas Evindar, Robert A. Batey · The Journal of Organic Chemistry · 2006 · 482 citations

Natural Sciences, Chemistry, Medicinal Chemistry +17

Ligand-Free Copper-Catalyzed Synthesis of Substituted Benzimidazoles, 2-Aminobenzimidazoles, 2-Aminobenzothiazoles, and Benzoxazoles

Prasenjit Saha, Ramana Tamminana, Nibadita Purkait et al. · The Journal of Organic Chemistry · 2009 · 347 citations

Natural Sciences, Chemical Engineering, Chemistry +14

Molecular Shape and Medicinal Chemistry: A Perspective

Anthony Nicholls, Georgia B. McGaughey, Robert P. Sheridan et al. · Journal of Medicinal Chemistry · 2010 · 313 citations · Full text

Pharmacy, Chemistry, Medicinal Chemistry +17