Life SciencesBiochemistryPharmacologyDrug DiscoveryEnzymologyProtein BiochemistryEnzyme InhibitionPeptide ChemistryPeptide Drug DiscoveryProtein ChemistryProtein StructureProteolytic EnzymesChemical Structure-activity RelationshipsProtease InhibitionProtease InhibitorsProtease SelectivitySerine Protease Mechanism
There are many compounds inhibiting serine proteases which play an important role in the human organism. This article reviews publications on the low-molecular weight, serine protease inhibitory cyanopeptides and reports on new developments in establishing structure-activity relationships.