Concepedia

The Synthesis of Novel Thiazole Containing Cyclic Peptides <i>via</i> Cyclooligomerisation Reactions

Anna Bertram, Katrina A. Jolliffe, Felix González-López de Turiso, Gerald Pattenden

Synlett · 1999 · 32 citations · 2 references

Concepts

Natural SciencesChemistryMedicinal ChemistryDrug DiscoveryOrganic ChemistryHeterocycle SynthesisHeterocyclic ChemistryHeterocyclic CompoundsOrganic SynthesisPeptide Bond ChemistryPeptide ChemistryAmino Acid-derived HeterocyclesCyclic PeptidesCyclized PeptidesCycloaddition ReactionsCyclopeptide SynthesisPeptide CyclizationThiazole ChemistryThiazole Synthesis

Abstract

Thiazole containing cyclic peptides have been synthesised in high yields by cyclooligomerisation reactions of amino acid substituted thiazole monomers.

References

2

A Novel Synthesis of Chiral 1-Allyl-1,2,3,4-tetrahydro-β-carboline Employing Allyltributyltin and Chiral Acyl Chlorides

Takashi Itoh, Yûji Matsuya, Yasuko Enomoto et al. · Synlett · 1999 · 20 citations

Natural Sciences, Chemistry, Drug Discovery +10

A New Method for the Synthesis of 5-Fluorouracil Prodrugs

Pascale Jolimaître, Christiane André‐Barrès, Myriam Malet‐Martino et al. · Synlett · 1999 · 12 citations

Pharmacy, Chemistry, Medicinal Chemistry +7