Concepedia

Synthesis of 2-aryl and coumarin substituted benzothiazole derivatives

Rajesh S. Kenny, Uday C. Mashelkar

Journal of Heterocyclic Chemistry · 2006 · 15 citations · 28 references

DOI

Concepts

Abstract

A facile and effective method for the synthesis of some benzothiazole derivatives is described. The method involves the action of aryl aldehyde and o-aminothiophenol in acetic acid resulting into in situ formation of the thiol substituted Schiff's base and its cyclization to 2-aryl benzothiazole upon prolonged heating.

References

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