Concepedia

(R)-[18F]NEBIFQUINIDE: A promising new PET tracer for TSPO imaging

Neydher Berroterán-Infante, Thomas Kalina, L. Fetty, Victoria Janisch, Ramona Velasco, Chrysoula Vraka, Marcus Hacker, Alexander Haug, Katharina Pallitsch, Wolfgang Wadsak,

European Journal of Medicinal Chemistry · 2019 · 18 citations · 20 references

DOI

Concepts

References

20

Relationship between the inhibition constant (KI) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction

Yung-Chi Cheng, William H. Prusoff · Biochemical Pharmacology · 1973 · 12.9K citations

, , +14

Specific benzodiazepine receptors in rat brain characterized by high-affinity (3H)diazepam binding.

Richard F. Squires · Proceedings of the National Academy of Sciences · 1977 · 1.3K citations · Full text

, , +12

An 18-kDa Translocator Protein (TSPO) Polymorphism Explains Differences in Binding Affinity of the PET Radioligand PBR28

David R. Owen, Astrid Yeo, Roger N. Gunn et al. · Journal of Cerebral Blood Flow & Metabolism · 2011 · 778 citations · Full text

, , +17

Mixed-Affinity Binding in Humans with 18-kDa Translocator Protein Ligands

David R. Owen, Roger N. Gunn, Eugenii A. Rabiner et al. · Journal of Nuclear Medicine · 2010 · 354 citations · Full text

, , +13

Radiosynthesis and initial evaluation of [18F]-FEPPA for PET imaging of peripheral benzodiazepine receptors

Alan A. Wilson, Armando García, Jun Parkes et al. · Nuclear Medicine and Biology · 2008 · 207 citations

, , +15