Concepedia

Cu-mediated synthesis of differentially substituted diazepines as AChE inhibitors; validation through molecular docking and Lipinski’s filter to develop novel anti-neurodegenerative drugs

N. Sudhapriya, Manish Kumar, Paramasivan T. Perumal

Bioorganic & Medicinal Chemistry Letters · 2019 · 33 citations · 30 references

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References

30

The maximal affinity of ligands

Irwin D. Kuntz, K. Chen, Kim A. Sharp et al. · Proceedings of the National Academy of Sciences · 1999 · 840 citations

Opium alkaloid noscapine is an antitumor agent that arrests metaphase and induces apoptosis in dividing cells

Keqiang Ye, Yong Ke, Nagalakshmi Keshava et al. · Proceedings of the National Academy of Sciences · 1998 · 342 citations · Full text

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Novel bioactive isoquinoline alkaloids from Carduus crispus

Qingying Zhang, Guangzhong Tu, Yuying Zhao et al. · Tetrahedron · 2002 · 234 citations

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6-Phenyl-4H-s-triazolo[4,3-a][1,4]benzodiazepines which have central nervous system depressant activity

Jackson B. Hester, Allan D. Rudzik, Bharat V. Kamdar · Journal of Medicinal Chemistry · 1971 · 211 citations

, , +19

Enantioselective Double Manipulation of Tetrahydroisoquinolines with Terminal Alkynes and Aldehydes under Copper(I) Catalysis

Weilong Lin, Tao Cao, Fan Wu et al. · Angewandte Chemie International Edition · 2013 · 159 citations