Peptide conjugates of lactoferricin analogues and antimicrobials—Design, chemical synthesis, and evaluation of antimicrobial activity and mammalian cytotoxicity

A Stepwise Huisgen Cycloaddition Process: Copper(I)-Catalyzed Regioselective “Ligation” of Azides and Terminal Alkynes

Vsevolod V. Rostovtsev, Luke G. Green, Valery V. Fokin et al. · Angewandte Chemie International Edition · 2002 · 11.5K citations

Natural Sciences, Chemistry, Catalysis +8

Peptidotriazoles on Solid Phase:  [1,2,3]-Triazoles by Regiospecific Copper(I)-Catalyzed 1,3-Dipolar Cycloadditions of Terminal Alkynes to Azides

Christian W. Tornøe, Caspar Christensen, Morten Meldal · The Journal of Organic Chemistry · 2002 · 8.5K citations

Pharmacy, Medicinal Chemistry, Catalysis +12

Peptoids: a modular approach to drug discovery.

Reyna J. Simon, Robert S. Kania, Ronald N. Zuckermann et al. · Proceedings of the National Academy of Sciences · 1992 · 941 citations

Pharmacy, Biochemistry, Molecular Biology +17

Identification of the bactericidal domain of lactoferrin

Wayne Bellamy, Mitsunori Takase, Koji Yamauchi et al. · Biochimica et Biophysica Acta (BBA) - Protein Structure and Molecular Enzymology · 1992 · 890 citations

Life Sciences, Microbiology, Molecular Biology +6

<em>Ex Vivo</em> Red Blood Cell Hemolysis Assay for the Evaluation of pH-responsive Endosomolytic Agents for Cytosolic Delivery of Biomacromolecular Drugs

Brian C. Evans, Christopher E. Nelson, Shann S. Yu et al. · Journal of Visualized Experiments · 2013 · 356 citations · Full text

Pharmacy, Pharmaceutics, Pharmacology +13