Organic Process Research & Development · 2019 · 28 citations · 29 references
Natural SciencesChemical EngineeringChemistryGreen ChemistryNatural Product BiosynthesisOrganic ChemistryHeterocycle SynthesisHeterocyclic ChemistryHigh-throughput SynthesisMacrocycle SynthesisMicrowave-assisted SynthesisOrganic SynthesisContinuous FlowContinuous Flow ProcessingFlow-based High-throughput SynthesisMacrocycle Library SynthesisMacrocyclic Library SynthesisMicrowave-assisted Cyclization ReactionsOlefin MetathesisOlefin Metathesis Catalysis
The renewable macrocyclic musk 3-methylcyclohexadec-6-enone was prepared via macrocyclic olefin metathesis on gram scale using two different protocols: a room temperature batch process which afforded a 57% yield of the desired macrocycle, but required long reaction times (5 d). In contrast, a continuous flow strategy provided a lower yield of 32% of macrocycle, although the short reaction times (150 °C, 5 min) improve throughput (1 g/4.8 h). Batch and continuous flow protocols were also tested on other macrocyclizations involving substrates bearing trisubstituted olefins.
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