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CYP enzymes, expressed within live human suspension cells, are superior to widely-used microsomal enzymes in identifying potent CYP1A1/CYP1B1 inhibitors: Identification of quinazolinones as CYP1A1/CYP1B1 inhibitors that efficiently reverse B[a]P toxicity and cisplatin resistance
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Citations
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References
2019
Year
Cisplatin ResistanceCyp1a1/cyp1b1 InhibitorsDrug TargetMedicineCyp EnzymesAnti-cancer AgentDrug DevelopmentPharmacologyCell BiologyDrug DiscoveryDrug Resistance
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